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Teisinis statusas
Patentas neįsigaliojo (pagal EPK)
| (51) | INT.CL. | C07D 487/18 | (2006.01) |
| A61P 35/00 | (2006.01) | ||
| A61P 3/10 | (2006.01) | ||
| A61P 17/06 | (2006.01) | ||
| A61P 19/02 | (2006.01) | ||
| A61P 19/06 | (2006.01) | ||
| A61P 19/10 | (2006.01) | ||
| A61P 25/16 | (2006.01) | ||
| A61P 25/28 | (2006.01) | ||
| A61K 31/415 | (2006.01) |
| (11) | Patento numeris | 3253764 |
| (13) | Dokumento rūšis | T |
| (96) | Europos patento paraiškos numeris | 16706472.4 |
| Europos patento paraiškos padavimo data | 2016-02-05 | |
| (97) | Europos patento paraiškos paskelbimo data | 2017-12-13 |
| (45) | Paskelbimo apie Europos patento išdavimą data | 2021-06-09 |
| (46) | Apibrėžties vertimo paskelbimo data |
| (86) | Numeris | PCT/US2016/016709 |
| Data | 2016-02-05 |
| (87) | Numeris | WO 2016/127025 |
| Data | 2016-08-11 |
| (30) | Numeris | Data | Šalis |
| 201562112374 P | 2015-02-05 | US |
| (72) |
CHEN, Xiaoling , US
YU, Henry , US
LAN, Ruoxi , US
JORAND-LEBRUN, Catherine , US
JOHNSON, Theresa L. , US
GOUTOPOULOS, Andreas , US
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| (73) |
Merck Patent GmbH ,
Frankfurter Strasse 250, 64293 Darmstadt,
DE
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| (54) | MACROCYCLIC COMPOUNDS AS IRAK1/4 INHIBITORS AND USES THEREOF |
| MACROCYCLIC COMPOUNDS AS IRAK1/4 INHIBITORS AND USES THEREOF |