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(51) | INT.CL. | C07H 19/207 | (2013.01) |
C07H 19/10 | (2006.01) | ||
C07H 19/24 | (2006.01) | ||
C07H 19/044 | (2013.01) | ||
A61P 31/14 | (2018.01) | ||
C07H 19/207 | (2006.01) | ||
C07H 19/04 | (2013.01) | ||
C07H 19/20 | (2006.01) | ||
C07F 9/65586 | (2013.01) | ||
C07H 19/06 | (2006.01) | ||
C07H 19/052 | (2006.01) | ||
C07H 19/24 | (2013.01) | ||
C07H 19/10 | (2013.01) | ||
A61K 31/7072 | (2006.01) | ||
A61P 31/00 | (2018.01) | ||
A61P 31/14 | (2006.01) | ||
C07F 9/65517 | (2013.01) | ||
C07H 19/044 | (2006.01) | ||
C07F 9/65616 | (2013.01) | ||
C07F 9/22 | (2006.01) | ||
C07F 7/1804 | (2013.01) | ||
C07H 19/04 | (2006.01) | ||
C07H 19/06 | (2013.01) | ||
A61K 31/664 | (2006.01) | ||
C07F 9/2458 | (2013.01) | ||
A61K 31/716 | (2006.01) | ||
C07F 9/242 | (2013.01) | ||
C07F 7/18 | (2006.01) | ||
C07H 19/20 | (2013.01) | ||
C07F 9/6558 | (2006.01) | ||
C07H 19/052 | (2013.01) | ||
C07F 9/24 | (2006.01) | ||
C07F 9/655 | (2006.01) | ||
C07F 9/6561 | (2006.01) | ||
A61P 31/00 | (2006.01) |
(11) | Number of the document | 3290428 |
(13) | Kind of document | T |
(96) | European patent application number | 17172585.6 |
Date of filing the European patent application | 2011-03-31 | |
(97) | Date of publication of the European application | 2018-03-07 |
(45) | Date of publication and mention of the grant of the patent | 2021-10-13 |
(46) | Date of publication of the claims translation |
(30) | Number | Date | Country code |
319513 P | 2010-03-31 | US | |
319548 P | 2010-03-31 | US | |
783680 | 2010-05-20 | US |
(72) |
Ross, Bruce S , US
Sofia, Michael Joseph , US
Pamulapati, Ganapati Reddy , US
Rachakonda, Suguna , US
Zhang, Hai-Ren , US
Chun, Byoung-Kwon , US
Wang, Peiyuan , US
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(73) |
Gilead Pharmasset LLC ,
c/o Gilead Sciences, Inc.
333 Lakeside Drive, Foster City, CA 94404,
US
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(54) | TABLET COMPRISING CRYSTALLINE (S)-ISOPROPYL 2-(((S)-(((2R,3R,4R,5R)-5-(2,4-DIOXO-3,4-DIHYDROPYRIMIDIN-1 (2H)-YL)-4-FLUORO-3-HYDROXY-4-METHYLTETRAHYDROFURAN-2-YL)METHOXY)(PHENOXY)PHOSPHORYL)AMINO)PROPANOATE |
TABLET COMPRISING CRYSTALLINE (S)-ISOPROPYL 2-(((S)-(((2R,3R,4R,5R)-5-(2,4-DIOXO-3,4-DIHYDROPYRIMIDIN-1 (2H)-YL)-4-FLUORO-3-HYDROXY-4-METHYLTETRAHYDROFURAN-2-YL)METHOXY)(PHENOXY)PHOSPHORYL)AMINO)PROPANOATE |