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EN | LT
LT - TABLET COMPRISING CRYSTALLINE (S)-ISOPROPYL 2-(((S)-(((2R,3R,4R,5R)-5-(2,4-DIOXO-3,4-DIHYDROPYRIMIDIN-1 (2H)-YL)-4-FLUORO-3-HYDROXY-4-METHYLTETRAHYDROFURAN-2-YL)METHOXY)(PHENOXY)PHOSPHORYL)AMINO)PROPANOATE
EN - TABLET COMPRISING CRYSTALLINE (S)-ISOPROPYL 2-(((S)-(((2R,3R,4R,5R)-5-(2,4-DIOXO-3,4-DIHYDROPYRIMIDIN-1 (2H)-YL)-4-FLUORO-3-HYDROXY-4-METHYLTETRAHYDROFURAN-2-YL)METHOXY)(PHENOXY)PHOSPHORYL)AMINO)PROPANOATE

Teisinis statusas

Patentas neįsigaliojo (pagal EPK)

Bibliografiniai duomenys
Tarptautinės patentų klasifikacijos indeksai (TPK)
(51) INT.CL. C07H 19/207 (2013.01)
C07H 19/10 (2006.01)
C07H 19/24 (2006.01)
C07H 19/044 (2013.01)
A61P 31/14 (2018.01)
C07H 19/207 (2006.01)
C07H 19/04 (2013.01)
C07H 19/20 (2006.01)
C07F 9/65586 (2013.01)
C07H 19/06 (2006.01)
C07H 19/052 (2006.01)
C07H 19/24 (2013.01)
C07H 19/10 (2013.01)
A61K 31/7072 (2006.01)
A61P 31/00 (2018.01)
A61P 31/14 (2006.01)
C07F 9/65517 (2013.01)
C07H 19/044 (2006.01)
C07F 9/65616 (2013.01)
C07F 9/22 (2006.01)
C07F 7/1804 (2013.01)
C07H 19/04 (2006.01)
C07H 19/06 (2013.01)
A61K 31/664 (2006.01)
C07F 9/2458 (2013.01)
A61K 31/716 (2006.01)
C07F 9/242 (2013.01)
C07F 7/18 (2006.01)
C07H 19/20 (2013.01)
C07F 9/6558 (2006.01)
C07H 19/052 (2013.01)
C07F 9/24 (2006.01)
C07F 9/655 (2006.01)
C07F 9/6561 (2006.01)
A61P 31/00 (2006.01)
Europos patentas
(11) Patento numeris 3290428
(13) Dokumento rūšis T
(96) Europos patento paraiškos numeris 17172585.6
Europos patento paraiškos padavimo data 2011-03-31
(97) Europos patento paraiškos paskelbimo data 2018-03-07
(45) Paskelbimo apie Europos patento išdavimą data 2021-10-13
(46) Apibrėžties vertimo paskelbimo data
Prioriteto paraiškos
(30) Numeris Data Šalis
319513 P 2010-03-31 US
319548 P 2010-03-31 US
783680 2010-05-20 US
Išradėjai
(72)
Ross, Bruce S , US
Sofia, Michael Joseph , US
Pamulapati, Ganapati Reddy , US
Rachakonda, Suguna , US
Zhang, Hai-Ren , US
Chun, Byoung-Kwon , US
Wang, Peiyuan , US
Savininkas
(73) Gilead Pharmasset LLC , c/o Gilead Sciences, Inc. 333 Lakeside Drive, Foster City, CA 94404, US
Pavadinimas
(54) TABLET COMPRISING CRYSTALLINE (S)-ISOPROPYL 2-(((S)-(((2R,3R,4R,5R)-5-(2,4-DIOXO-3,4-DIHYDROPYRIMIDIN-1 (2H)-YL)-4-FLUORO-3-HYDROXY-4-METHYLTETRAHYDROFURAN-2-YL)METHOXY)(PHENOXY)PHOSPHORYL)AMINO)PROPANOATE
  TABLET COMPRISING CRYSTALLINE (S)-ISOPROPYL 2-(((S)-(((2R,3R,4R,5R)-5-(2,4-DIOXO-3,4-DIHYDROPYRIMIDIN-1 (2H)-YL)-4-FLUORO-3-HYDROXY-4-METHYLTETRAHYDROFURAN-2-YL)METHOXY)(PHENOXY)PHOSPHORYL)AMINO)PROPANOATE