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LT - HYDROXYALKYLAMINE- AND HYDROXYCYCLOALKYLAMINE-SUBSTITUTED DIAMINE-ARYLSULFONAMIDE COMPOUNDS WITH SELECTIVE ACTIVITY IN VOLTAGE-GATED SODIUM CHANNELS
EN - HYDROXYALKYLAMINE- AND HYDROXYCYCLOALKYLAMINE-SUBSTITUTED DIAMINE-ARYLSULFONAMIDE COMPOUNDS WITH SELECTIVE ACTIVITY IN VOLTAGE-GATED SODIUM CHANNELS

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Patent not validated

Bibliographic data
Indications of the International Patent Classification (IPC)
(51) INT.CL. C07D 285/08
C07D 417/12
C07D 277/52
A61K 31/4168
A61K 31/4178
A61K 31/4196
A61K 31/551
A61P 29/00
A61P 11/14
European patent
(11) Number of the document 3390374
(13) Kind of document T
(96) European patent application number 16820497.2
Date of filing the European patent application 2016-12-14
(97) Date of publication of the European application 2018-10-24
(45) Date of publication and mention of the grant of the patent 2020-08-26
(46) Date of publication of the claims translation
PCT application
(86) Number PCT/US2016/066445
Date 2016-12-14
PCT application publication
(87) Number WO 2017/106226
Date 2017-06-22
Priority applications
(30) Number Date Country code
201562269327 P 2015-12-18 US
201662290235 P 2016-02-02 US
201662420956 P 2016-11-11 US
Inventors
(72)
GRESHOCK, Thomas, J., US
MULHEARN, James, US
ZHENG, Junying, US
KIM, Ronald, M., US
ZHANG, Ting, US
ROECKER, Anthony, J., US
WON, Walter, US
NANTERMET, Philippe, US
ANAND, Rajan, US
ZHOU, Gang, US
WANG, Deping, US
GUO, Liangqin, US
Grantee
(73) Merck Sharp & Dohme Corp., 126 East Lincoln Avenue, Rahway, NJ 07065-0907, US
Title
(54) HYDROXYALKYLAMINE- AND HYDROXYCYCLOALKYLAMINE-SUBSTITUTED DIAMINE-ARYLSULFONAMIDE COMPOUNDS WITH SELECTIVE ACTIVITY IN VOLTAGE-GATED SODIUM CHANNELS
  HYDROXYALKYLAMINE- AND HYDROXYCYCLOALKYLAMINE-SUBSTITUTED DIAMINE-ARYLSULFONAMIDE COMPOUNDS WITH SELECTIVE ACTIVITY IN VOLTAGE-GATED SODIUM CHANNELS