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LT - HYDROXYALKYLAMINE- AND HYDROXYCYCLOALKYLAMINE-SUBSTITUTED DIAMINE-ARYLSULFONAMIDE COMPOUNDS WITH SELECTIVE ACTIVITY IN VOLTAGE-GATED SODIUM CHANNELS
EN - HYDROXYALKYLAMINE- AND HYDROXYCYCLOALKYLAMINE-SUBSTITUTED DIAMINE-ARYLSULFONAMIDE COMPOUNDS WITH SELECTIVE ACTIVITY IN VOLTAGE-GATED SODIUM CHANNELS

Teisinis statusas

Patentas neįsigaliojo (pagal EPK)

Bibliografiniai duomenys
Tarptautinės patentų klasifikacijos indeksai (TPK)
(51) INT.CL. C07D 285/08
C07D 417/12
C07D 277/52
A61K 31/4168
A61K 31/4178
A61K 31/4196
A61K 31/551
A61P 29/00
A61P 11/14
Europos patentas
(11) Patento numeris 3390374
(13) Dokumento rūšis T
(96) Europos patento paraiškos numeris 16820497.2
Europos patento paraiškos padavimo data 2016-12-14
(97) Europos patento paraiškos paskelbimo data 2018-10-24
(45) Paskelbimo apie Europos patento išdavimą data 2020-08-26
(46) Apibrėžties vertimo paskelbimo data
Tarptautinės paraiškos padavimo
(86) Numeris PCT/US2016/066445
Data 2016-12-14
Tarptautinės paraiškos paskelbimo
(87) Numeris WO 2017/106226
Data 2017-06-22
Prioriteto paraiškos
(30) Numeris Data Šalis
201562269327 P 2015-12-18 US
201662290235 P 2016-02-02 US
201662420956 P 2016-11-11 US
Išradėjai
(72)
GRESHOCK, Thomas, J., US
MULHEARN, James, US
ZHENG, Junying, US
KIM, Ronald, M., US
ZHANG, Ting, US
ROECKER, Anthony, J., US
WON, Walter, US
NANTERMET, Philippe, US
ANAND, Rajan, US
ZHOU, Gang, US
WANG, Deping, US
GUO, Liangqin, US
Savininkas
(73) Merck Sharp & Dohme Corp., 126 East Lincoln Avenue, Rahway, NJ 07065-0907, US
Pavadinimas
(54) HYDROXYALKYLAMINE- AND HYDROXYCYCLOALKYLAMINE-SUBSTITUTED DIAMINE-ARYLSULFONAMIDE COMPOUNDS WITH SELECTIVE ACTIVITY IN VOLTAGE-GATED SODIUM CHANNELS
  HYDROXYALKYLAMINE- AND HYDROXYCYCLOALKYLAMINE-SUBSTITUTED DIAMINE-ARYLSULFONAMIDE COMPOUNDS WITH SELECTIVE ACTIVITY IN VOLTAGE-GATED SODIUM CHANNELS