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Teisinis statusas
Patentas neįsigaliojo (pagal EPK)
(51) | INT.CL. | C07D 241/18 | (2006.01) |
C07D 403/12 | (2013.01) | ||
C07D 241/20 | (2006.01) | ||
C07D 403/04 | (2013.01) | ||
C07D 403/12 | (2006.01) | ||
C07D 241/18 | (2013.01) | ||
C07D 403/04 | (2006.01) | ||
C07D 241/20 | (2013.01) | ||
A61K 31/497 | (2006.01) | ||
A61P 35/02 | (2018.01) | ||
A61K 31/4985 | (2006.01) | ||
A61P 35/04 | (2018.01) | ||
A61P 35/00 | (2006.01) | ||
C07D 401/04 | (2013.01) | ||
C07D 477/26 | (2013.01) | ||
C07D 487/04 | (2013.01) |
(11) | Patento numeris | 3484856 |
(13) | Dokumento rūšis | T |
(96) | Europos patento paraiškos numeris | 17742609.5 |
Europos patento paraiškos padavimo data | 2017-07-11 | |
(97) | Europos patento paraiškos paskelbimo data | 2019-05-22 |
(45) | Paskelbimo apie Europos patento išdavimą data | 2023-11-15 |
(46) | Apibrėžties vertimo paskelbimo data |
(86) | Numeris | PCT/US2017/041577 |
Data | 2017-07-11 |
(87) | Numeris | WO 2018/013597 |
Data | 2018-01-18 |
(30) | Numeris | Data | Šalis |
201662361249 P | 2016-07-12 | US | |
201762449523 P | 2017-01-23 | US |
(72) |
JOGALEKAR, Ashutosh , US
WON, Walter , US
KOLTUN, Elena S. , US
GILL, Adrian , US
MELLEM, Kevin , US
AAY, Naing , US
BUCKL, Andreas , US
SEMKO, Christopher , US
KISS, Gert , US
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(73) |
Revolution Medicines, Inc. ,
700 Saginaw Drive, Redwood City, CA 94063,
US
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(54) | 2,5-DISUBSTITUTED 3-METHYL PYRAZINES AND 2,5,6-TRISUBSTITUTED 3-METHYL PYRAZINES AS ALLOSTERIC SHP2 INHIBITORS |
2,5-DISUBSTITUTED 3-METHYL PYRAZINES AND 2,5,6-TRISUBSTITUTED 3-METHYL PYRAZINES AS ALLOSTERIC SHP2 INHIBITORS |