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Teisinis statusas
Patentas neįsigaliojo (pagal EPK)
| (51) | INT.CL. | A61K 31/5365 | (2013.01) | 
| C07D 207/456 | (2006.01) | ||
| C07D 403/14 | (2006.01) | ||
| A61K 47/68 | (2017.08) | ||
| C07D 401/14 | (2006.01) | ||
| A61P 35/00 | (2018.01) | ||
| C07D 491/18 | (2006.01) | ||
| C07D 207/456 | (2013.01) | ||
| C07D 519/00 | (2006.01) | ||
| C07D 401/14 | (2013.01) | ||
| C07K 5/027 | (2006.01) | ||
| C07D 403/14 | (2013.01) | ||
| C07K 7/02 | (2006.01) | ||
| C07D 491/18 | (2013.01) | ||
| A61K 47/68 | (2017.01) | ||
| C07D 519/00 | (2013.01) | ||
| C07K 7/02 | (2013.01) | ||
| A61K 31/5365 | (2006.01) | ||
| A61P 35/00 | (2006.01) | 
| (11) | Patento numeris | 3546448 | 
| (13) | Dokumento rūšis | T | 
| (96) | Europos patento paraiškos numeris | 17873634.4 | 
| Europos patento paraiškos padavimo data | 2017-11-24 | |
| (97) | Europos patento paraiškos paskelbimo data | 2019-10-02 | 
| (45) | Paskelbimo apie Europos patento išdavimą data | 2022-04-06 | 
| (46) | Apibrėžties vertimo paskelbimo data | 
| (86) | Numeris | PCT/CN2017/112958 | 
| Data | 2017-11-24 | 
| (87) | Numeris | WO 2018/095422 | 
| Data | 2018-05-31 | 
| (30) | Numeris | Data | Šalis | 
| 201611093699 | 2016-11-25 | CN | |
| 201711169847 | 2017-11-22 | CN | 
| (72) | 
                    
                    
                    
                    
                    SHEN, Jingkang , CN  
                    
                    
                    
                    
                    MENG, Tao , CN  
                    
                    
                    
                    
                    MA, Lanping , CN  
                    
                    
                    
                    
                    WANG, Xin , CN  
                    
                    
                    
                    
                    PENG, Hongli , CN  
                    
                    
                    
                    
                    ZHANG, Yongliang , CN  
                    
                    
                    
                    
                    YU, Ting , CN  
                    
                    
                    
                    
                    CHEN, Lin , CN  
                    
                    
                    
                    
                    DU, Zhiyan , CN  
                    
                    
                    
                    
                    WANG, Ying , CN  | 
| (73) | Mabwell (Shanghai) Bioscience Co., Ltd. ,
                Building 3 
No.576 Libing Road, Pudong New Area
Shanghai,
                CN Jiangsu Mabwell Health Pharmaceutical R&D Co., Ltd. , 3F, National New Drug Innovation Base 1 Avenue, China Medical City Taizhou Jiangsu, CN | 
| (54) | DI-SUBSTITUTED MALEIC AMIDE LINKER FOR ANTIBODY-DRUG CONJUGATING AND PREPARATION METHOD AND USE THEREOF | 
| DI-SUBSTITUTED MALEIC AMIDE LINKER FOR ANTIBODY-DRUG CONJUGATING AND PREPARATION METHOD AND USE THEREOF |