|
|
Legal status
Patent not validated
| (51) | INT.CL. | C07D 471/04 | (2006.01) |
| C07D 471/04 | (2013.01) | ||
| C07D 519/00 | (2006.01) | ||
| C07D 519/00 | (2013.01) |
| (11) | Number of the document | 3694853 |
| (13) | Kind of document | T |
| (96) | European patent application number | 18796238.6 |
| Date of filing the European patent application | 2018-10-10 | |
| (97) | Date of publication of the European application | 2020-08-19 |
| (45) | Date of publication and mention of the grant of the patent | 2023-05-17 |
| (46) | Date of publication of the claims translation |
| (86) | Number | PCT/US2018/055255 |
| Date | 2018-10-10 |
| (87) | Number | WO 2019/075092 |
| Date | 2019-04-18 |
| (30) | Number | Date | Country code |
| 201762570565 P | 2017-10-10 | US |
| (72) |
EARY, Charles Todd , US
SPENCER, Stacey , US
CRANE, Zack , US
CHANDO, Katelyn , US
ASSELIN, Sylvie , US
LIU, Weidong , US
WELCH, Mike , US
COOK, Adam , US
KOLAKOWSKI, Gabrielle R. , US
METCALF, Andrew T. , US
MORENO, David A. , US
TANG, Tony P. , US
|
| (73) |
Array BioPharma Inc. ,
3200 Walnut Street, Boulder, CO 80301,
US
Loxo Oncology, Inc. , Lilly Corporate Centre Indianapolis, Indiana 46285, US |
| (54) | PROCESS FOR THE PREPARATION OF 6-(2-HYDROXY-2-METHYLPROPOXY)-4-(6-(6-((6-METHOXYPYRIDIN-3-YL)METHYL)-3,6-DIAZABICYCLO[3.1.1]HEPTAN-3-YL)PYRIDIN-3-YL)PYRAZOLO[1,5-A]PYRIDINE-3-CARBONITRILE |
| PROCESS FOR THE PREPARATION OF 6-(2-HYDROXY-2-METHYLPROPOXY)-4-(6-(6-((6-METHOXYPYRIDIN-3-YL)METHYL)-3,6-DIAZABICYCLO[3.1.1]HEPTAN-3-YL)PYRIDIN-3-YL)PYRAZOLO[1,5-A]PYRIDINE-3-CARBONITRILE |