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Teisinis statusas
Patentas neįsigaliojo (pagal EPK)
| (51) | INT.CL. | C07D 471/04 | (2006.01) |
| C07D 471/04 | (2013.01) | ||
| C07D 519/00 | (2006.01) | ||
| C07D 519/00 | (2013.01) |
| (11) | Patento numeris | 3694853 |
| (13) | Dokumento rūšis | T |
| (96) | Europos patento paraiškos numeris | 18796238.6 |
| Europos patento paraiškos padavimo data | 2018-10-10 | |
| (97) | Europos patento paraiškos paskelbimo data | 2020-08-19 |
| (45) | Paskelbimo apie Europos patento išdavimą data | 2023-05-17 |
| (46) | Apibrėžties vertimo paskelbimo data |
| (86) | Numeris | PCT/US2018/055255 |
| Data | 2018-10-10 |
| (87) | Numeris | WO 2019/075092 |
| Data | 2019-04-18 |
| (30) | Numeris | Data | Šalis |
| 201762570565 P | 2017-10-10 | US |
| (72) |
EARY, Charles Todd , US
SPENCER, Stacey , US
CRANE, Zack , US
CHANDO, Katelyn , US
ASSELIN, Sylvie , US
LIU, Weidong , US
WELCH, Mike , US
COOK, Adam , US
KOLAKOWSKI, Gabrielle R. , US
METCALF, Andrew T. , US
MORENO, David A. , US
TANG, Tony P. , US
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| (73) |
Array BioPharma Inc. ,
3200 Walnut Street, Boulder, CO 80301,
US
Loxo Oncology, Inc. , Lilly Corporate Centre Indianapolis, Indiana 46285, US |
| (54) | PROCESS FOR THE PREPARATION OF 6-(2-HYDROXY-2-METHYLPROPOXY)-4-(6-(6-((6-METHOXYPYRIDIN-3-YL)METHYL)-3,6-DIAZABICYCLO[3.1.1]HEPTAN-3-YL)PYRIDIN-3-YL)PYRAZOLO[1,5-A]PYRIDINE-3-CARBONITRILE |
| PROCESS FOR THE PREPARATION OF 6-(2-HYDROXY-2-METHYLPROPOXY)-4-(6-(6-((6-METHOXYPYRIDIN-3-YL)METHYL)-3,6-DIAZABICYCLO[3.1.1]HEPTAN-3-YL)PYRIDIN-3-YL)PYRAZOLO[1,5-A]PYRIDINE-3-CARBONITRILE |