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LT - PROCESS FOR THE PREPARATION OF 6-(2-HYDROXY-2-METHYLPROPOXY)-4-(6-(6-((6-METHOXYPYRIDIN-3-YL)METHYL)-3,6-DIAZABICYCLO[3.1.1]HEPTAN-3-YL)PYRIDIN-3-YL)PYRAZOLO[1,5-A]PYRIDINE-3-CARBONITRILE
EN - PROCESS FOR THE PREPARATION OF 6-(2-HYDROXY-2-METHYLPROPOXY)-4-(6-(6-((6-METHOXYPYRIDIN-3-YL)METHYL)-3,6-DIAZABICYCLO[3.1.1]HEPTAN-3-YL)PYRIDIN-3-YL)PYRAZOLO[1,5-A]PYRIDINE-3-CARBONITRILE

Teisinis statusas

Patentas neįsigaliojo (pagal EPK)

Bibliografiniai duomenys
Tarptautinės patentų klasifikacijos indeksai (TPK)
(51) INT.CL. C07D 471/04 (2006.01)
C07D 471/04 (2013.01)
C07D 519/00 (2006.01)
C07D 519/00 (2013.01)
Europos patentas
(11) Patento numeris 3694853
(13) Dokumento rūšis T
(96) Europos patento paraiškos numeris 18796238.6
Europos patento paraiškos padavimo data 2018-10-10
(97) Europos patento paraiškos paskelbimo data 2020-08-19
(45) Paskelbimo apie Europos patento išdavimą data 2023-05-17
(46) Apibrėžties vertimo paskelbimo data
Tarptautinės paraiškos padavimo
(86) Numeris PCT/US2018/055255
Data 2018-10-10
Tarptautinės paraiškos paskelbimo
(87) Numeris WO 2019/075092
Data 2019-04-18
Prioriteto paraiškos
(30) Numeris Data Šalis
201762570565 P 2017-10-10 US
Išradėjai
(72)
EARY, Charles Todd , US
SPENCER, Stacey , US
CRANE, Zack , US
CHANDO, Katelyn , US
ASSELIN, Sylvie , US
LIU, Weidong , US
WELCH, Mike , US
COOK, Adam , US
KOLAKOWSKI, Gabrielle R. , US
METCALF, Andrew T. , US
MORENO, David A. , US
TANG, Tony P. , US
Savininkas
(73) Array BioPharma Inc. , 3200 Walnut Street, Boulder, CO 80301, US
Loxo Oncology, Inc. , Lilly Corporate Centre Indianapolis, Indiana 46285, US
Pavadinimas
(54) PROCESS FOR THE PREPARATION OF 6-(2-HYDROXY-2-METHYLPROPOXY)-4-(6-(6-((6-METHOXYPYRIDIN-3-YL)METHYL)-3,6-DIAZABICYCLO[3.1.1]HEPTAN-3-YL)PYRIDIN-3-YL)PYRAZOLO[1,5-A]PYRIDINE-3-CARBONITRILE
  PROCESS FOR THE PREPARATION OF 6-(2-HYDROXY-2-METHYLPROPOXY)-4-(6-(6-((6-METHOXYPYRIDIN-3-YL)METHYL)-3,6-DIAZABICYCLO[3.1.1]HEPTAN-3-YL)PYRIDIN-3-YL)PYRAZOLO[1,5-A]PYRIDINE-3-CARBONITRILE