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LT - IMPROVED METHOD FOR THE MANUFACTURE OF 3-[(1S)-1-IMIDAZO[1,2-A]PYRIDIN-6-YLETHYL]-5-(1-METHYLPYRAZOL-4-YL)TRIAZOLO[4,5-B]PYRAZINE AND POLYMORPHIC FORMS THEREOF
EN - IMPROVED METHOD FOR THE MANUFACTURE OF 3-[(1S)-1-IMIDAZO[1,2-A]PYRIDIN-6-YLETHYL]-5-(1-METHYLPYRAZOL-4-YL)TRIAZOLO[4,5-B]PYRAZINE AND POLYMORPHIC FORMS THEREOF

Teisinis statusas

Patentas neįsigaliojo (pagal EPK)

Bibliografiniai duomenys
Tarptautinės patentų klasifikacijos indeksai (TPK)
(51) INT.CL. C07D 471/04 (2006.01)
C07D 519/00 (2013.01)
C07D 519/00 (2006.01)
C07D 471/04 (2013.01)
Europos patentas
(11) Patento numeris 3849977
(13) Dokumento rūšis T
(96) Europos patento paraiškos numeris 19769738.6
Europos patento paraiškos padavimo data 2019-09-10
(97) Europos patento paraiškos paskelbimo data 2021-07-21
(45) Paskelbimo apie Europos patento išdavimą data 2023-07-19
(46) Apibrėžties vertimo paskelbimo data
Tarptautinės paraiškos padavimo
(86) Numeris PCT/EP2019/074083
Data 2019-09-10
Tarptautinės paraiškos paskelbimo
(87) Numeris WO 2020/053198
Data 2020-03-19
Prioriteto paraiškos
(30) Numeris Data Šalis
PCT/CN2018/104941 2018-09-11 WO
Išradėjai
(72)
TURNER, Andrew, Roy , GB
TURNER, Andrew, Timothy , GB
HOWELL, Gareth, Paul , GB
GALL, Malcolm, Allan, Young , GB
MULHOLLAND, Keith, Raymond , GB
ADLINGTON, Neil, Keith , GB
TIAN, Zhenping , CN
LIU, Bo , CN
GONG, Qisun , CN
YU, Wei , CN
Savininkas
(73) Astrazeneca AB , 151 85 Södertälje, SE
Hutchison Medipharma Limited , Building 4 720 Cai Lun Road Pilot Free Zone, Shanghai 201203, CN
Pavadinimas
(54) IMPROVED METHOD FOR THE MANUFACTURE OF 3-[(1S)-1-IMIDAZO[1,2-A]PYRIDIN-6-YLETHYL]-5-(1-METHYLPYRAZOL-4-YL)TRIAZOLO[4,5-B]PYRAZINE AND POLYMORPHIC FORMS THEREOF
  IMPROVED METHOD FOR THE MANUFACTURE OF 3-[(1S)-1-IMIDAZO[1,2-A]PYRIDIN-6-YLETHYL]-5-(1-METHYLPYRAZOL-4-YL)TRIAZOLO[4,5-B]PYRAZINE AND POLYMORPHIC FORMS THEREOF