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EN | LT
LT - NOVEL SYNTHETIC OPTIONS TOWARDS THE MANUFACTURE OF (6R,10S)-10- {4-[5-CHLORO-2-(4-CHLORO-1H-1,2,3-TRIAZOL-1-YL)PHENYL]-6-OXO-1(6H)- PYRIMIDINYL}- 1-(DIFLUOROMETHYL)-6-METHYL-1,4,7,8,9,10-HEXAHYDRO-11,15 -(METHENO)PYRAZOLO [4,3-B] [1,7] DIAZACYCLOTETRADECIN-5(6H)-ONE
EN - NOVEL SYNTHETIC OPTIONS TOWARDS THE MANUFACTURE OF (6R,10S)-10- {4-[5-CHLORO-2-(4-CHLORO-1H-1,2,3-TRIAZOL-1-YL)PHENYL]-6-OXO-1(6H)- PYRIMIDINYL}- 1-(DIFLUOROMETHYL)-6-METHYL-1,4,7,8,9,10-HEXAHYDRO-11,15 -(METHENO)PYRAZOLO [4,3-B] [1,7] DIAZACYCLOTETRADECIN-5(6H)-ONE

Teisinis statusas

Patentas neįsigaliojo (pagal EPK)

Bibliografiniai duomenys
Tarptautinės patentų klasifikacijos indeksai (TPK)
(51) INT.CL. C07D 213/61 (2006.01)
C07D 471/18 (2013.01)
C07D 401/04 (2006.01)
C07D 213/61 (2013.01)
C07D 471/18 (2006.01)
C07D 401/04 (2013.01)
Europos patentas
(11) Patento numeris 3953334
(13) Dokumento rūšis T
(96) Europos patento paraiškos numeris 20721374.5
Europos patento paraiškos padavimo data 2020-04-10
(97) Europos patento paraiškos paskelbimo data 2022-02-16
(45) Paskelbimo apie Europos patento išdavimą data 2023-11-22
(46) Apibrėžties vertimo paskelbimo data
Tarptautinės paraiškos padavimo
(86) Numeris PCT/US2020/027655
Data 2020-04-10
Tarptautinės paraiškos paskelbimo
(87) Numeris WO 2020/210613
Data 2020-10-15
Prioriteto paraiškos
(30) Numeris Data Šalis
201962832614 P 2019-04-11 US
Išradėjai
(72)
CUNIERE, Nicolas , US
FAN, Yu , US
KOLOTUCHIN, Sergei , US
MUKHERJEE, Subha , US
SIMMONS, Eric M. , US
SINGH, Amarjit , US
WEI, Carolyn S. , US
XIAO, Yi , US
YUAN, Changxia , US
ZHENG, Bin , US
WAGSCHAL, Simon Albert , CH
BROGGINI, Diego Fernando Domenico , CH
CAO, Duy Chi Trung , CH
CHERNICHENKO, Kostiantyn , BE
LEMAIRE, Sébastien François Emmanuel , BE
BEN HAIM, Cyril , BE
Savininkas
(73) Bristol-Myers Squibb Company , Route 206 and Province Line Road, Princeton, NJ 08543, US
Janssen Pharmaceutica NV , Turnhoutseweg 30, 2340 Beerse, BE
Pavadinimas
(54) NOVEL SYNTHETIC OPTIONS TOWARDS THE MANUFACTURE OF (6R,10S)-10- {4-[5-CHLORO-2-(4-CHLORO-1H-1,2,3-TRIAZOL-1-YL)PHENYL]-6-OXO-1(6H)- PYRIMIDINYL}- 1-(DIFLUOROMETHYL)-6-METHYL-1,4,7,8,9,10-HEXAHYDRO-11,15 -(METHENO)PYRAZOLO [4,3-B] [1,7] DIAZACYCLOTETRADECIN-5(6H)-ONE
  NOVEL SYNTHETIC OPTIONS TOWARDS THE MANUFACTURE OF (6R,10S)-10- {4-[5-CHLORO-2-(4-CHLORO-1H-1,2,3-TRIAZOL-1-YL)PHENYL]-6-OXO-1(6H)- PYRIMIDINYL}- 1-(DIFLUOROMETHYL)-6-METHYL-1,4,7,8,9,10-HEXAHYDRO-11,15 -(METHENO)PYRAZOLO [4,3-B] [1,7] DIAZACYCLOTETRADECIN-5(6H)-ONE