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Teisinis statusas
Patentas neįsigaliojo (pagal EPK)
(51) | INT.CL. | C07D 213/61 | (2006.01) |
C07D 471/18 | (2013.01) | ||
C07D 401/04 | (2006.01) | ||
C07D 213/61 | (2013.01) | ||
C07D 471/18 | (2006.01) | ||
C07D 401/04 | (2013.01) |
(11) | Patento numeris | 3953334 |
(13) | Dokumento rūšis | T |
(96) | Europos patento paraiškos numeris | 20721374.5 |
Europos patento paraiškos padavimo data | 2020-04-10 | |
(97) | Europos patento paraiškos paskelbimo data | 2022-02-16 |
(45) | Paskelbimo apie Europos patento išdavimą data | 2023-11-22 |
(46) | Apibrėžties vertimo paskelbimo data |
(86) | Numeris | PCT/US2020/027655 |
Data | 2020-04-10 |
(87) | Numeris | WO 2020/210613 |
Data | 2020-10-15 |
(30) | Numeris | Data | Šalis |
201962832614 P | 2019-04-11 | US |
(72) |
CUNIERE, Nicolas , US
FAN, Yu , US
KOLOTUCHIN, Sergei , US
MUKHERJEE, Subha , US
SIMMONS, Eric M. , US
SINGH, Amarjit , US
WEI, Carolyn S. , US
XIAO, Yi , US
YUAN, Changxia , US
ZHENG, Bin , US
WAGSCHAL, Simon Albert , CH
BROGGINI, Diego Fernando Domenico , CH
CAO, Duy Chi Trung , CH
CHERNICHENKO, Kostiantyn , BE
LEMAIRE, Sébastien François Emmanuel , BE
BEN HAIM, Cyril , BE
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(73) |
Bristol-Myers Squibb Company ,
Route 206 and Province Line Road, Princeton, NJ 08543,
US
Janssen Pharmaceutica NV , Turnhoutseweg 30, 2340 Beerse, BE |
(54) | NOVEL SYNTHETIC OPTIONS TOWARDS THE MANUFACTURE OF (6R,10S)-10- {4-[5-CHLORO-2-(4-CHLORO-1H-1,2,3-TRIAZOL-1-YL)PHENYL]-6-OXO-1(6H)- PYRIMIDINYL}- 1-(DIFLUOROMETHYL)-6-METHYL-1,4,7,8,9,10-HEXAHYDRO-11,15 -(METHENO)PYRAZOLO [4,3-B] [1,7] DIAZACYCLOTETRADECIN-5(6H)-ONE |
NOVEL SYNTHETIC OPTIONS TOWARDS THE MANUFACTURE OF (6R,10S)-10- {4-[5-CHLORO-2-(4-CHLORO-1H-1,2,3-TRIAZOL-1-YL)PHENYL]-6-OXO-1(6H)- PYRIMIDINYL}- 1-(DIFLUOROMETHYL)-6-METHYL-1,4,7,8,9,10-HEXAHYDRO-11,15 -(METHENO)PYRAZOLO [4,3-B] [1,7] DIAZACYCLOTETRADECIN-5(6H)-ONE |