LT - PROCESSES AND INTERMEDIATES FOR THE PREPARATION OF 2-(2,6-DICHLOROPHENYL)-1-[(1S,3R)-3-(HYDROXYMETHYL)-5-(3-HYDROXY-3-METHYLBUTYL)-1-METHYL-3,4-DIHYDROISOQUINOLIN-2(1H)-YL]ETHENONE
EN - PROCESSES AND INTERMEDIATES FOR THE PREPARATION OF 2-(2,6-DICHLOROPHENYL)-1-[(1S,3R)-3-(HYDROXYMETHYL)-5-(3-HYDROXY-3-METHYLBUTYL)-1-METHYL-3,4-DIHYDROISOQUINOLIN-2(1H)-YL]ETHENONE
Legal status
Patent not validated
Bibliographic data
Indications of the International Patent Classification (IPC)
| (51) |
INT.CL. |
C07D 217/16 |
(2006.01) |
|
|
C07D 217/16 |
(2013.01) |
|
|
C07D 263/24 |
(2006.01) |
|
|
C07D 263/24 |
(2013.01) |
|
|
C07D 498/04 |
(2006.01) |
|
|
C07D 498/04 |
(2013.01) |
European patent
| (11) |
Number of the document |
3986867 |
| (13) |
Kind of document |
T |
| (96) |
European patent application number |
20751718.6 |
|
Date of filing the European patent application |
2020-06-11 |
| (97) |
Date of publication of the European application |
2022-04-27 |
| (45) |
Date of publication and mention of the grant of the patent |
2023-09-13
|
| (46) |
Date of publication of the claims translation |
|
PCT application
| (86) |
Number |
PCT/US2020/037186 |
|
Date |
2020-06-11 |
PCT application publication
| (87) |
Number |
WO 2020/257043 |
|
Date |
2020-12-24 |
Priority applications
| (30) |
Number |
Date |
Country code |
|
201962862805 P |
2019-06-18
|
US |
Inventors
| (72) |
COLE, Kevin Paul , US
KALLMAN, Neil John , US
MAGNUS, Nicholas Andrew , US
|
Grantee
| (73) |
ELI LILLY AND COMPANY ,
Lilly Corporate Center, Indianapolis, IN 46206-6288,
US
|
Title
| (54) |
PROCESSES AND INTERMEDIATES FOR THE PREPARATION OF 2-(2,6-DICHLOROPHENYL)-1-[(1S,3R)-3-(HYDROXYMETHYL)-5-(3-HYDROXY-3-METHYLBUTYL)-1-METHYL-3,4-DIHYDROISOQUINOLIN-2(1H)-YL]ETHENONE |
| |
PROCESSES AND INTERMEDIATES FOR THE PREPARATION OF 2-(2,6-DICHLOROPHENYL)-1-[(1S,3R)-3-(HYDROXYMETHYL)-5-(3-HYDROXY-3-METHYLBUTYL)-1-METHYL-3,4-DIHYDROISOQUINOLIN-2(1H)-YL]ETHENONE |
