LT - PROCESSES AND INTERMEDIATES FOR THE PREPARATION OF 2-(2,6-DICHLOROPHENYL)-1-[(1S,3R)-3-(HYDROXYMETHYL)-5-(3-HYDROXY-3-METHYLBUTYL)-1-METHYL-3,4-DIHYDROISOQUINOLIN-2(1H)-YL]ETHENONE
EN - PROCESSES AND INTERMEDIATES FOR THE PREPARATION OF 2-(2,6-DICHLOROPHENYL)-1-[(1S,3R)-3-(HYDROXYMETHYL)-5-(3-HYDROXY-3-METHYLBUTYL)-1-METHYL-3,4-DIHYDROISOQUINOLIN-2(1H)-YL]ETHENONE
Teisinis statusas
Patentas neįsigaliojo (pagal EPK)
Bibliografiniai duomenys
Tarptautinės patentų klasifikacijos indeksai (TPK)
(51) |
INT.CL. |
C07D 217/16 |
(2006.01) |
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C07D 217/16 |
(2013.01) |
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C07D 263/24 |
(2006.01) |
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C07D 263/24 |
(2013.01) |
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C07D 498/04 |
(2006.01) |
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C07D 498/04 |
(2013.01) |
Europos patentas
(11) |
Patento numeris |
3986867 |
(13) |
Dokumento rūšis |
T |
(96) |
Europos patento paraiškos numeris |
20751718.6 |
|
Europos patento paraiškos padavimo data |
2020-06-11 |
(97) |
Europos patento paraiškos paskelbimo data |
2022-04-27 |
(45) |
Paskelbimo apie Europos patento išdavimą data |
2023-09-13
|
(46) |
Apibrėžties vertimo paskelbimo data |
|
Tarptautinės paraiškos padavimo
(86) |
Numeris |
PCT/US2020/037186 |
|
Data |
2020-06-11 |
Tarptautinės paraiškos paskelbimo
(87) |
Numeris |
WO 2020/257043 |
|
Data |
2020-12-24 |
Prioriteto paraiškos
(30) |
Numeris |
Data |
Šalis |
|
201962862805 P |
2019-06-18
|
US |
Išradėjai
(72) |
COLE, Kevin Paul , US
KALLMAN, Neil John , US
MAGNUS, Nicholas Andrew , US
|
Savininkas
(73) |
ELI LILLY AND COMPANY ,
Lilly Corporate Center, Indianapolis, IN 46206-6288,
US
|
Pavadinimas
(54) |
PROCESSES AND INTERMEDIATES FOR THE PREPARATION OF 2-(2,6-DICHLOROPHENYL)-1-[(1S,3R)-3-(HYDROXYMETHYL)-5-(3-HYDROXY-3-METHYLBUTYL)-1-METHYL-3,4-DIHYDROISOQUINOLIN-2(1H)-YL]ETHENONE |
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PROCESSES AND INTERMEDIATES FOR THE PREPARATION OF 2-(2,6-DICHLOROPHENYL)-1-[(1S,3R)-3-(HYDROXYMETHYL)-5-(3-HYDROXY-3-METHYLBUTYL)-1-METHYL-3,4-DIHYDROISOQUINOLIN-2(1H)-YL]ETHENONE |