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EN | LT
LT - PROCESSES AND INTERMEDIATES FOR THE PREPARATION OF 2-(2,6-DICHLOROPHENYL)-1-[(1S,3R)-3-(HYDROXYMETHYL)-5-(3-HYDROXY-3-METHYLBUTYL)-1-METHYL-3,4-DIHYDROISOQUINOLIN-2(1H)-YL]ETHENONE
EN - PROCESSES AND INTERMEDIATES FOR THE PREPARATION OF 2-(2,6-DICHLOROPHENYL)-1-[(1S,3R)-3-(HYDROXYMETHYL)-5-(3-HYDROXY-3-METHYLBUTYL)-1-METHYL-3,4-DIHYDROISOQUINOLIN-2(1H)-YL]ETHENONE

Teisinis statusas

Patentas neįsigaliojo (pagal EPK)

Bibliografiniai duomenys
Tarptautinės patentų klasifikacijos indeksai (TPK)
(51) INT.CL. C07D 217/16 (2006.01)
C07D 217/16 (2013.01)
C07D 263/24 (2006.01)
C07D 263/24 (2013.01)
C07D 498/04 (2006.01)
C07D 498/04 (2013.01)
Europos patentas
(11) Patento numeris 3986867
(13) Dokumento rūšis T
(96) Europos patento paraiškos numeris 20751718.6
Europos patento paraiškos padavimo data 2020-06-11
(97) Europos patento paraiškos paskelbimo data 2022-04-27
(45) Paskelbimo apie Europos patento išdavimą data 2023-09-13
(46) Apibrėžties vertimo paskelbimo data
Tarptautinės paraiškos padavimo
(86) Numeris PCT/US2020/037186
Data 2020-06-11
Tarptautinės paraiškos paskelbimo
(87) Numeris WO 2020/257043
Data 2020-12-24
Prioriteto paraiškos
(30) Numeris Data Šalis
201962862805 P 2019-06-18 US
Išradėjai
(72)
COLE, Kevin Paul , US
KALLMAN, Neil John , US
MAGNUS, Nicholas Andrew , US
Savininkas
(73) ELI LILLY AND COMPANY , Lilly Corporate Center, Indianapolis, IN 46206-6288, US
Pavadinimas
(54) PROCESSES AND INTERMEDIATES FOR THE PREPARATION OF 2-(2,6-DICHLOROPHENYL)-1-[(1S,3R)-3-(HYDROXYMETHYL)-5-(3-HYDROXY-3-METHYLBUTYL)-1-METHYL-3,4-DIHYDROISOQUINOLIN-2(1H)-YL]ETHENONE
  PROCESSES AND INTERMEDIATES FOR THE PREPARATION OF 2-(2,6-DICHLOROPHENYL)-1-[(1S,3R)-3-(HYDROXYMETHYL)-5-(3-HYDROXY-3-METHYLBUTYL)-1-METHYL-3,4-DIHYDROISOQUINOLIN-2(1H)-YL]ETHENONE