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LT - N-((1,2,3,5,6,7-HEXAHYDRO-S-INDACEN-4-YL)CARBAMOYL)-4,5,6,7-TETRAHYDROBENZOFURAN-2-SULFONAMIDE DERIVATIVES AND RELATED COMPOUNDS AS NLPR3 MODULATORS FOR THE TREATMENT OF MULTIPLE SCLEROSIS (MS)
EN - N-((1,2,3,5,6,7-HEXAHYDRO-S-INDACEN-4-YL)CARBAMOYL)-4,5,6,7-TETRAHYDROBENZOFURAN-2-SULFONAMIDE DERIVATIVES AND RELATED COMPOUNDS AS NLPR3 MODULATORS FOR THE TREATMENT OF MULTIPLE SCLEROSIS (MS)

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Bibliographic data
Indications of the International Patent Classification (IPC)
(51) INT.CL. C07D 307/82 (2013.01)
C07D 307/82 (2006.01)
C07D 491/04 (2006.01)
C07D 491/04 (2013.01)
A61P 3/00 (2018.01)
C07D 333/62 (2006.01)
C07C 311/56 (2006.01)
A61P 3/04 (2018.01)
A61K 31/343 (2006.01)
A61P 3/10 (2018.01)
A61K 31/55 (2006.01)
A61P 1/04 (2018.01)
A61K 31/4162 (2006.01)
A61P 1/16 (2018.01)
A61P 1/04 (2006.01)
A61P 11/00 (2018.01)
A61P 1/16 (2006.01)
A61P 11/06 (2018.01)
A61P 25/28 (2018.01)
A61P 3/00 (2006.01)
A61P 37/00 (2018.01)
A61P 3/04 (2006.01)
A61P 37/06 (2018.01)
A61P 3/10 (2006.01)
A61P 9/00 (2018.01)
A61P 9/00 (2006.01)
A61P 9/10 (2018.01)
A61P 9/10 (2006.01)
C07D 333/62 (2013.01)
A61P 11/00 (2006.01)
A61P 11/06 (2006.01)
A61P 25/28 (2006.01)
A61P 37/00 (2006.01)
A61P 37/06 (2006.01)
European patent
(11) Number of the document 3999496
(13) Kind of document T
(96) European patent application number 20757941.8
Date of filing the European patent application 2020-07-16
(97) Date of publication of the European application 2022-05-25
(45) Date of publication and mention of the grant of the patent 2024-12-18
(46) Date of publication of the claims translation
PCT application
(86) Number PCT/IB2020/000634
Date 2020-07-16
PCT application publication
(87) Number WO 2021/009566
Date 2021-01-21
Priority applications
(30) Number Date Country code
201962875402 P 2019-07-17 US
Inventors
(72)
MOHAN, Raju , US
NUSS, John , US
HARRIS, Jason , US
YUAN, Shendong , US
Grantee
(73) Zomagen Biosciences Ltd , 662 Encinitas Blvd., Suite 250, Encinitas, CA 92024, US
Title
(54) N-((1,2,3,5,6,7-HEXAHYDRO-S-INDACEN-4-YL)CARBAMOYL)-4,5,6,7-TETRAHYDROBENZOFURAN-2-SULFONAMIDE DERIVATIVES AND RELATED COMPOUNDS AS NLPR3 MODULATORS FOR THE TREATMENT OF MULTIPLE SCLEROSIS (MS)
  N-((1,2,3,5,6,7-HEXAHYDRO-S-INDACEN-4-YL)CARBAMOYL)-4,5,6,7-TETRAHYDROBENZOFURAN-2-SULFONAMIDE DERIVATIVES AND RELATED COMPOUNDS AS NLPR3 MODULATORS FOR THE TREATMENT OF MULTIPLE SCLEROSIS (MS)