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LT - N-((1,2,3,5,6,7-HEXAHYDRO-S-INDACEN-4-YL)CARBAMOYL)-4,5,6,7-TETRAHYDROBENZOFURAN-2-SULFONAMIDE DERIVATIVES AND RELATED COMPOUNDS AS NLPR3 MODULATORS FOR THE TREATMENT OF MULTIPLE SCLEROSIS (MS)
EN - N-((1,2,3,5,6,7-HEXAHYDRO-S-INDACEN-4-YL)CARBAMOYL)-4,5,6,7-TETRAHYDROBENZOFURAN-2-SULFONAMIDE DERIVATIVES AND RELATED COMPOUNDS AS NLPR3 MODULATORS FOR THE TREATMENT OF MULTIPLE SCLEROSIS (MS)

Teisinis statusas

Patentas neįsigaliojo (pagal EPK)

Bibliografiniai duomenys
Tarptautinės patentų klasifikacijos indeksai (TPK)
(51) INT.CL. C07D 307/82 (2013.01)
C07D 307/82 (2006.01)
C07D 491/04 (2006.01)
C07D 491/04 (2013.01)
A61P 3/00 (2018.01)
C07D 333/62 (2006.01)
C07C 311/56 (2006.01)
A61P 3/04 (2018.01)
A61K 31/343 (2006.01)
A61P 3/10 (2018.01)
A61K 31/55 (2006.01)
A61P 1/04 (2018.01)
A61K 31/4162 (2006.01)
A61P 1/16 (2018.01)
A61P 1/04 (2006.01)
A61P 11/00 (2018.01)
A61P 1/16 (2006.01)
A61P 11/06 (2018.01)
A61P 25/28 (2018.01)
A61P 3/00 (2006.01)
A61P 37/00 (2018.01)
A61P 3/04 (2006.01)
A61P 37/06 (2018.01)
A61P 3/10 (2006.01)
A61P 9/00 (2018.01)
A61P 9/00 (2006.01)
A61P 9/10 (2018.01)
A61P 9/10 (2006.01)
C07D 333/62 (2013.01)
A61P 11/00 (2006.01)
A61P 11/06 (2006.01)
A61P 25/28 (2006.01)
A61P 37/00 (2006.01)
A61P 37/06 (2006.01)
Europos patentas
(11) Patento numeris 3999496
(13) Dokumento rūšis T
(96) Europos patento paraiškos numeris 20757941.8
Europos patento paraiškos padavimo data 2020-07-16
(97) Europos patento paraiškos paskelbimo data 2022-05-25
(45) Paskelbimo apie Europos patento išdavimą data 2024-12-18
(46) Apibrėžties vertimo paskelbimo data
Tarptautinės paraiškos padavimo
(86) Numeris PCT/IB2020/000634
Data 2020-07-16
Tarptautinės paraiškos paskelbimo
(87) Numeris WO 2021/009566
Data 2021-01-21
Prioriteto paraiškos
(30) Numeris Data Šalis
201962875402 P 2019-07-17 US
Išradėjai
(72)
MOHAN, Raju , US
NUSS, John , US
HARRIS, Jason , US
YUAN, Shendong , US
Savininkas
(73) Zomagen Biosciences Ltd , 662 Encinitas Blvd., Suite 250, Encinitas, CA 92024, US
Pavadinimas
(54) N-((1,2,3,5,6,7-HEXAHYDRO-S-INDACEN-4-YL)CARBAMOYL)-4,5,6,7-TETRAHYDROBENZOFURAN-2-SULFONAMIDE DERIVATIVES AND RELATED COMPOUNDS AS NLPR3 MODULATORS FOR THE TREATMENT OF MULTIPLE SCLEROSIS (MS)
  N-((1,2,3,5,6,7-HEXAHYDRO-S-INDACEN-4-YL)CARBAMOYL)-4,5,6,7-TETRAHYDROBENZOFURAN-2-SULFONAMIDE DERIVATIVES AND RELATED COMPOUNDS AS NLPR3 MODULATORS FOR THE TREATMENT OF MULTIPLE SCLEROSIS (MS)