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Teisinis statusas
Patentas galioja
| (51) | INT.CL. | C07D 471/04 | (2006.01) |
| C07D 498/04 | (2006.01) | ||
| A61K 31/522 | (2006.01) | ||
| A61P 35/00 | (2006.01) |
| (11) | Patento numeris | 4051678 |
| (13) | Dokumento rūšis | T |
| (96) | Europos patento paraiškos numeris | 20815976.4 |
| Europos patento paraiškos padavimo data | 2020-10-27 | |
| (97) | Europos patento paraiškos paskelbimo data | 2022-09-07 |
| (45) | Paskelbimo apie Europos patento išdavimą data | 2026-03-04 |
| (46) | Apibrėžties vertimo paskelbimo data | 2026-05-11 |
| (86) | Numeris | PCT/US2020/057496 |
| Data | 2020-10-27 |
| (87) | Numeris | WO 2021/086833 |
| Data | 2021-05-06 |
| (30) | Numeris | Data | Šalis |
| 201962926879 P | 2019-10-28 | US | |
| 202063030014 P | 2020-05-26 | US |
| (72) |
BHARATHAN, Indu , US
GATHIAKA, Symon , US
GRAHAM, Thomas, H. , US
HAN, Yongxin , US
HENDERSON, Timothy , US
HENNESSY, Elisabeth , US
MA, Xiaoshen , US
OTTE, Ryan , US
PALANI, Anandan , US
SLOMAN, David, L. , US
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| (73) |
Merck Sharp & Dohme LLC ,
126 East Lincoln Avenue
P.O. Box 2000, Rahway, New Jersey 07065,
US
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| (74) |
Reda ŽABOLIENĖ,
METIDA, Verslo centras "VERTAS", Gynėjų g. 16, LT-01109 Vilnius,
LT
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| (54) | Mažamolekuliniai KRAS G12C mutanto inhibitoriai |
| SMALL MOLECULE INHIBITORS OF KRAS G12C MUTANT |